DMPX
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| Clinical data | |
|---|---|
| ATC code | none |
| Identifiers | |
| CAS Number |
14114-46-6  Y |
| PubChem (CID) | 99562 |
| ChemSpider | 89948 |
| ECHA InfoCard | 100.162.258 |
| Chemical and physical data | |
| Formula | C10H10N4O2 |
| Molar mass | 218.212 g/mol |
| 3D model (Jmol) | Interactive image |
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DMPX (3,7-Dimethyl-1-propargylxanthine) is a caffeine analog which displays affinity to A2-adenosine receptors, in contrast to the A1 subtype receptors.[1] DMPX had 28× & 15× higher potency than caffeine in blocking peripheral and central NECA-responses. The locomotor stimulation caused by DMPX (ED50 10 μmol/kg) was similarly higher than caffeine.[1]
See also
- DPCPX
- 8-PT
- CPX (8-CPT)
- 8-Chlorotheophylline
- Theophylline
References
- 1 2 3,7-Dimethyl-1-propargylxanthine: a potent and selective in vivo antagonist of adenosine analogs. Life Sci. 1988;43(21):1671-84. PMID 3193854
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